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dicyclomine - medtigo

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dicyclomine

Brand Name :

Bentyl

Synonyms :

dicyclomine

Class :

Anticholinergic agents





No data available for drug.

Actions and Spectrum: 

dicyclomine is a medication that belongs to the class of anticholinergic drugs, and it acts on the smooth muscles of the gastrointestinal (GI) tract. The actions and spectrum of dicyclomine can be summarized as follows: 

  • Antispasmodic effects: dicyclomine works by blocking the action of acetylcholine at muscarinic receptors in the smooth muscles of the GI tract, which leads to relaxation of the muscles and a decrease in spasms. This makes it useful in the treatment of conditions that involve abdominal pain and cramping, such as irritable bowel syndrome (IBS). 
  • Anti-secretory effects: dicyclomine can also reduce the secretion of gastric acid, which can be helpful in the treatment of peptic ulcers. 
  • Local anesthetic effects: dicyclomine has some local anesthetic effects on the GI tract, which can help to reduce pain and discomfort associated with GI spasms. 

The spectrum of dicyclomine includes its use in the treatment of various GI disorders, such as IBS, functional bowel disorders, diverticulitis, and peptic ulcers. dicyclomine is often used in combination with other medications, such as proton pump inhibitors (PPIs), to provide a comprehensive approach to the management of GI disorders. It is important to note that dicyclomine is a prescription medication and should only be used under the guidance of a healthcare professional. 

DRUG INTERACTION

dicyclomine

&

  • prednisolone and gentamicin ophthalmic
  • promethazine and codeine
  • poractant alfa
  • protamine sulfate
  • aflibercept intravitreal
  • prednicarbate
  • promethazine/dextromethorphan
  • codeine, phenylephrine, and promethazine
  • potassium phosphate
  • glatiramer acetate
  • gentamicin (Ophthalmic)
  • leniolisib
  • rezafungin
  • fluorometholone
  • dalfampridine
  • hydrocortisone topical 
  • empagliflozin and linagliptin
  • triamcinolone topical
  • minocycline topical
  • minocycline dental
  • ketotifen ophthalmic
  • darunavir and cobicistat
  • lidocaine topical
  • neomycin/polymyxin B/bacitracin/lidocaine (OTC)
  • lidocaine/ hydrocortisone
  • lidocaine anesthetic
  • lidocaine ophthalmic
  • lidocaine/tetracaine
  • desonide
  • dabigatran
  • fexofenadine
  • fluoride
  • decitabine and cedazuridine
  • dasiglucagon
  • hydroxypropyl cellulose ophthalmic
  • epoetin alfa
  • ibritumomab tiuxetan
  • trimethobenzamide
  • dexamethasone/ tobramycin
  • tafasitamab
  • valacyclovir
  • mebendazole
  • levoleucovorin
  • flaxseed
  • germanium
  • glutathione
  • lycopene
  • pygeum
  • horseradish
  • ziv-aflibercept
  • micafungin
  • trofinetide
  • taliglucerase alfa
  • tildrakizumab
  • sulopenem (Pending FDA Approval)
  • thyrotropin alfa
  • birch
  • thrombin, topical
  • tivozanib
  • tafluprost
  • methohexital
  • urea and hydrocortisone
  • unoprostone ophthalmic
  • trihexyphenidyl
  • ezetimibe
  • evolocumab
  • trifluridine and tipiracil
  • methenamine
  • misoprostol
  • miltefosine
  • rimantadine
  • maralixibat
  • coenzyme Q10
  • chlorella
  • garlic
  • forskolin
  • zavegepant
  • menotropins
  • margetuximab
  • meprobamate
  • melarsoprol
  • evening primrose oil
  • lemongrass
  • molindone
  • fenugreek
  • phytosterols
  • red yeast rice
  • uridine triacetate
  • tropicamide
  • incobotulinumtoxinA
  • Grape Seed Extract
  • carbachol ophthalmic
  • cosyntropin
  • cyclopentolate and phenylephrine
  • carteolol ophthalmic
  • pentazocine/naloxone
  • pentazocine/acetaminophen
  • casimersen
  • carisoprodol, aspirin, and codeine
  • carisoprodol
  • carboprost tromethamine
  • flurandrenolide
  • brinzolamide/brimonidine
  • betamethasone topical
  • omaveloxolone
  • bardoxolone
  • allogeneic processed thymus tissue
  • fluocinolone topical
  • tacrolimus topical
  • ruxolitnib topical
  • pimecrolimus topical
  • sofosbuvir, velpatasvir and voxilaprevir
  • sofosbuvir/velpatasvir
  • mitotane
  • elbasvir/​grazoprevir
  • wheat dextrin
  • vanadium
  • iron/folic acid/vitamin/mineral
  • molybdenum
  • sparsentan
  • velmanase alfa-tycv
  • pegcetacoplan
  • ferrous sulfate
  • cyclosporine ophthalmic
  • ferric pyrophosphate
  • ammonium lactate
  • etelcalcetide
  • iodoquinol
  • sucroferric oxyhydroxide
  • doxercalciferol
  • terconazole vaginal
  • cortisone
  • pyronaridine
  • tetrahydrozoline, ophthalmic
  • tenapanor
  • tesamorelin
  • benazepril/hydrochlorothiazide
  • nadolol and bendroflumethiazide
  • spironolactone and hydrochlorothiazide
  • COVID-19 Vaccine, mRNA
  • atosiban
  • bisoprolol and hydrochlorothiazide
  • ephedrine/guaifenesin
  • clonidine/chlorthalidone
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  • amlodipine/valsartan/hydrochlorothiazide
  • hydrochlorothiazide and irbesartan
  • candesartan/hydrochlorothiazide
  • ciclesonide intranasal
  • cromolyn sodium ophthalmic
  • methyldopa/hydrochlorothiazide
  • valsartan/hydrochlorothiazide
  • hydrochlorothiazide and triamterene
  • moexipril/hydrochlorothiazide
  • mometasone/intranasal
  • ofloxacin ophthalmic
  • cysteamine
  • metoprolol/hydrochlorothiazide
  • amlodipine/olmesartan
  • eprosartan/hydrochlorothiazide
  • amlodipine/telmisartan
  • hydrochlorothiazide/aliskiren
  • betamethasone/clotrimazole
  • telmisartan/hydrochlorothiazide
  • benazepril/amlodipine
  • bezlotoxumab
  • propranolol/hydrochlorothiazide
  • bupropion/naltrexone
  • burosumab
  • acetylcholine chloride intraocular solution
  • bupivacaine and meloxicam
  • budesonide and formoterol (inhalation)
  • valerian
  • entacapone/levodopa/carbidopa
  • carbidopa/levodopa
  • calaspargase pegol
  • cabotegravir
  • cefixime
  • calfactant
  • brinzolamide
  • daprodustat
  • brimonidine and timolol
  • brodalumab
  • buprenorphine and naloxone
  • hydrocortisone acetic acid otic
  • butorphanol
  • butoconazole
  • adapalene and benzoyl peroxide
  • acrivastine and pseudoephedrine
  • neomycin/polymyxin B/bacitracin topical
  • midodrine
  • baloxavir marboxil
  • bacitracin, neomycin, polymyxin B, and hydrocortisone topical
  • avatrombopag
  • glucagon
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  • adefovir
  • activated charcoal
  • avalglucosidase alfa
  • aclidinium and formoterol
  • iclaprim (Pending FDA Approval)
  • ampicillin/sulbactam
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  • acetaminophen and caffeine
  • acetaminophen/pamabrom
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  • anifrolumab
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  • anidulafungin
  • acetohydroxamic acid
  • alogliptin/pioglitazone
  • anthralin
  • pirtobrutinib
  • gabapentin
  • galsulfase
  • gadoterate meglumine
  • ferric gluconate
  • ferric derisomaltose
  • ethanolamine oleate
  • eteplirsen
  • vasopressin
  • desmopressin
  • meropenem/vaborbactam
  • ecallantide
  • econazole topical
  • dornase alfa
  • aspirin/dipyridamole
  • dipyridamole
  • difenoxin and atropine
  • diflorasone
  • difluprednate ophthalmic
  • eptinezumab
  • diethylpropion
  • dexchlorpheniramine
  • dexmethylphenidate
  • serdexmethylphenidate/​dexmethylphenidate
  • bexagliflozin
  • galcanezumab
  • fremanezumab
  • tapinarof topical
  • darifenacin
  • dalbavancin
  • darbepoetin alfa
  • azilsartan
  • colestipol
  • corticorelin
  • crotamiton
  • crofelemer
  • allogeneic cultured keratinocytes/fibroblasts in bovine collagen
  • tapentadol
  • cyclopentolate
  • polymyxin B/bacitracin topical
  • ketoconazole topical
  • tavaborole
  • tagraxofusp
  • crisaborole
  • crizanlizumab
  • satralizumab
  • spinosad
  • sacubitril/valsartan
  • sargramostim
  • sebelipase alfa
  • regadenoson
  • ribociclib/letrozole
  • ragweed allergen extract
  • radium-223 dichloride
  • secnidazole
  • setmelanotide
  • polycarbophil
  • plecanatide
  • sacituzumab govitecan
  • pertuzumab
  • pertuzumab/trastuzumab/hyaluronidase
  • pamidronate
  • halcinonide
  • glecaprevir/​pibrentasvir
  • glucarpidase
  • golodirsen
  • dextrose
  • hexaminolevulinate
  • iohexol
  • ferric citrate
  • elapegademase
  • emicizumab
  • erenumab
  • danaparoid
  • dantrolene
  • eflapegrastim
  • edaravone
  • amcinonide
  • carglumic acid
  • alcaftadine ophthalmic
  • agalsidase beta
  • afamelanotide
  • fosdenopterin
  • lidocaine and chlorhexidine
  • levorphanol
  • calcifediol
  • factor VIIa, recombinant
  • triheptanoin
  • peanut oral allergen powder
  • teprotumumab
  • poly-L-lactic acid/carboxymethylcellulose/mannitol
  • xenon Xe 129 hyperpolarized
  • ublituximab
  • anacaulase
  • glatiramer
  • peginterferon beta-1a
  • interferon beta-1a
  • onabotulinumtoxinA
  • cycloserine
  • ethionamide
  • cabotegravir and rilpivirine
  • vericiguat
  • omidenepag isopropyl
  • azelastine/fluticasone intranasal
  • benzyl peroxide
  • vutrisiran
  • brimonidine
  • testosterone topical
  • lenacapavir
  • tebentafusp
  • mosunetuzumab
  • faricimab
  • ganirelix
  • nadofaragene firadenovec
  • ozenoxacin
  • guaifenesin
  • adagrasib
  • guselkumab
  • adalimumab-aacf
  • nonoxynol-9
  • nifurtimox
  • nusinersen
  • nitazoxanide
  • mavacamten
  • calcipotriene
  • bimatoprost
  • obinutuzumab
  • amifostine
  • oxycodone/​aspirin
  • oxycodone/ibuprofen
  • oteseconazole
  • oxychlorosene
  • porfimer
  • pramoxine /hydrocortisone topical
  • podofilox
  • quinapril/hydrochlorothiazide
  • acetaminophen/pamabrom/pyrilamine
  • levobunolol
  • paregoric
  • idursulfase
  • lesinurad and allopurinol
  • latanoprost/​netarsudil ophthalmic
  • lactase enzyme
  • bioadherent oral
  • latanoprost and timolol
  • latanoprostene bunod
  • ledipasvir/sofosbuvir
  • imipenem/cilastatin/relebactam
  • imipenem/cilastatin
  • hemin
  • deucravacitinib
  • house dust mite allergen extract
  • halobetasol topical/tazarotene
  • remimazolam
  • somatropin
  • remifentanil
  • ethotoin
  • etidronate
  • empagliflozin, linagliptin, and metformin
  • elvitegravir/cobicistat/emtricitabine/tenofovir AF
  • empagliflozin/​linagliptin
  • evinacumab
  • finasteride and tadalafil
  • flortaucipir (18F)
  • proparacaine/ fluorescein ophthalmic
  • fluorescein/benoxinate ophthalmic
  • fluphenazine
  • alogliptin/​metformin
  • alogliptin/pioglitazone
  • alitretinoin topical
  • dextrose/ sodium citrate/fructose
  • dasabuvir
  • ombitasvir​/paritaprevir/​ritonavir
  • hydrocodone/​chlorpheniramine/​pseudoephedrine
  • hydroxyamphetamine/​tropicamide
  • acamprosate
  • gadobutrol
  • teclistamab
  • tremelimumab
  • futibatinib
  • etranacogene dezaparvovec
  • olutasidenib
  • naproxen and diphenhydramine
  • naratriptan
  • gadopiclenol
  • gadoxetate
  • gadoversetamide
  • naphazoline/pheniramine
  • naphazoline
  • nalbuphine
  • vosoritide
  • vitamin K1 (phytonadione)
  • moxidectin
  • basiliximab
  • fecal microbiota, live-jslm
  • ibuprofen/famotidine
  • famotidine
  • raxibacumab
  • omalizumab
  • measles, mumps, rubella, and varicella vaccine, live (Rx)
  • senna/docusate
  • dinoprostone
  • measles mumps and rubella vaccine, live
  • immune globulin IM (IGIM)
  • dyclonine
  • doravirine, lamivudine, and tenofovir disoproxil fumarate
  • elexacaftor/tezacaftor/ivacaftor
  • ivacaftor/tezacaftor
  • treosulfan
  • tranexamic acid
  • norethindrone acetate/​estradiol/​elagolix
  • artesunate
  • trientine
  • trifarotene
  • ziconotide
  • vonoprazan/amoxicillin/clarithromycin
  • pyrithione zinc
  • zinc oxide topical
  • naphazoline/​zinc sulfate/​glycerin ophthalmic
  • voretigene neparvovec
  • nirmatrelvir/ritonavir
  • bebetelovimab
  • sodium chloride
  • relugolix/​estradiol/​norethindrone
  • defibrotide
  • prothionamide
  • liraglutide
  • maitake
  • etilfrine
  • alpha-lipoic acid
  • ramosetron
  • olodaterol/tritropium
  • cimetropium
  • umeclidinium
  • itopride
  • secretin
  • naftopidil
  • trimeprazine
  • benperidol
  • chlormethiazole
  • multivitamins
  • secukinumab
  • glycopyrrolate inhaled and formoterol
  • amitriptyline and chlordiazepoxide
  • tirzepatide
  • relugolix/estradiol/norethindrone
  • mupirocin
  • alvimopan
  • chlordiazepoxide
  • insulin regular human
  • insulin aspart protamine/​insulin aspart
  • insulin isophane human/​insulin regular human
  • insulin degludec/insulin aspart
  • teplizumab
  • chlordiazepoxide/clidinium
  • aspirin, sodium bicarbonate, and citric acid
  • aluminum hydroxide, magnesium hydroxide, and simethicone
  • glycopyrrolate inhaled
  • olodaterol/tiotropium
  • umeclidinium bromide
  • timolol/dorzolamide
  • travoprost ophthalmic
  • loxapine
  • eptifibatide
  • hydrocodone/acetaminophen
  • omega 3 fatty acids
  • trandolapril/​verapamil
  • abciximab
  • artificial saliva
  • diphtheria, hepatitis B, pertussis (acellular), polio, and tetanus vaccine
  • diphtheria, haemophilus B, pertussis, polio, tetanus vaccine
  • haemophilus influenzae type b vaccine/hepatitis b vaccine
  • butalbital/aspirin/caffeine 
  • colchicine/probenecid
  • atovaquone and proguanil
  • ursodiol
  • chenodiol
  • casirivimab/imdevimab
  • tixagevimab/cilgavimab
  • molnupiravir
  • bebtelovimab
  • calcium, magnesium, potassium and sodium oxybate
  • sodium oxybate
  • diphtheria, polio, pertussis acellular, tetanus vaccine
  • pseudoephedrine loratadine
  • sodium chloride nasal
  • hydroxychloroquine sulfate
  • atorvastatin and ezetimibe
  • teriparatide
  • alendronate and cholecalciferol
  • alprostadil (IV)
  • romosozumab
  • risedronate
  • alendronate
  • glyburide/metformin
  • clorazepate
  • rosuvastatin/​ezetimibe
  • paclitaxel/encequidar
  • valsartan/amlodipine
  • enalapril/hydrochlorothiazide
  • enalapril and felodipine
  • amiloride/hydrochlorothiazide
  • triamterene/hydrochlorothiazide
  • lisinopril/hydrochlorothiazide
  • tegaserod
  • rhein
  • ritanserin
  • sulfaphenazole
  • sulconazole
  • taurursodiol
  • bromeperidol
  • carbapenems
  • fotemustine
  • difelikefalin
  • bromopride
  • alizapride
  • olopatadine
  • oxomemazine
  • paraldehyde
  • oxcarbazepine
  • kratom
  • elexacaftor
  • oritavancin
  • miocamycin
  • curcumin sulfate
  • seproxetine
  • clotrimazole
  • remacemide
  • piperine
  • ditiocarb
  • danoprevir
  • oxetacaine
  • topiroxostat
  • indisulam
  • tofisopam
  • noscapine
  • thiopental
  • tioconazole
  • nicotinamide
  • rutin
  • mequitazine
  • somatostatin
  • vapreotide
  • econazole
  • saracatinib
  • lestaurtinib
  • efonidipine
  • zimelidine
  • indalpine
  • desvenlafaxine
  • benidipine
  • dapoxetine
  • tesmilifene
  • pergolide
  • sitaxentan
  • resveratrol
  • bifonazole
  • tildipirosin
  • solithromycin
  • selamectin
  • imiquimod topical
  • fluorouracil topical
  • peginterferon alfa-2b
  • interferon alfa-2b
  • alteplase
  • tanshinone I
  • rosmarinic acid
  • caryophyllene
  • ursolic acid
  • cepharanthine
  • veliflapon
  • mirikizumab
  • cp-96345
  • famprofazone
  • peoniflorin
  • fepradinol
  • licofelone
  • polmacoxib
  • ebselen
  • taxifolin
  • betulinic acid
  • flurbiprofen axetil
  • talniflumate
  • morniflumate
  • nitroaspirin
  • firocoxib
  • ns-398
  • cimicoxib
  • robenacoxib
  • sc-236
  • imidazole salicylate
  • trolamine salicylate
  • pirprofen
  • benorilate
  • ethenzamide
  • mofebutazone
  • proquazone
  • carbaspirin calcium
  • guacetisal
  • proglumetacin
  • propyphenazone
  • pranoprofen
  • bendazac
  • tenidap
  • lonazolac
  • nifenazone
  • flunoxaprofen
  • difenpiramide
  • feprazone
  • bufexamac
  • alminoprofen
  • suxibuzone
  • fentiazac
  • tinoridine
  • tepoxalin
  • indobufen
  • flunixin
  • propacetamol
  • clonixin
  • droxicam
  • epirizole
  • etofenamate
  • ibuproxam
  • indoprofen
  • kebuzone
  • felbinac
  • zaltoprofen
  • azapropazone
  • zomepirac
  • niflumic acid
  • magnesium salicylate
  • suprofen
  • nepafenac
  • bromfenac
  • ciprofloxacin and hydrocortisone (otic) (Rx)
  • hydrocortisone/neomycin/polymyxin otic (Rx)
  • vigabatrine
  • valproate
  • tezepelumab (Rx)
  • triamcinolone acetonide/nystatin
  • triamcinolone suprachoroidal (Rx)
  • triamcinolone, intranasal
  • ciclesonide inhaled
  • diosmin
  • tirbanibulin
  • padeliporfin
  • roxadustat
  • aminosalicylic acid
  • rasburicase
  • tetracaine
  • articaine
  • ropivacaine
  • nitrous oxide
  • sulfapyridine
  • sulfanilamide
  • mafenide
  • isometheptene
  • amyl nitrite
  • antipyrine
  • isosorbide dinitrate
  • prilocaine
  • nitroglycerin
  • tobacco
  • batefenterol
  • hexoprenaline
  • pf-00610355
  • racepinephrine
  • protokylol
  • doxofylline
  • phenylpropanolamine
  • isoetharine
  • ephedra sinica root
  • dipivefrin
  • arbutamine
  • norepinephrine
  • fenoterol
  • clenbuterol
  • pirbuterol
  • epinephrine
  • ritodrine
  • procaterol
  • orciprenaline
  • bitolterol
  • abediterol
  • fluticasone furoate, umeclidinium and vilanterol
  • fluticasone furoate and vilanterol
  • mometasone and formoterol
  • pramoxine topical (OTC)
  • menthol/pramoxine (topical)
  • tetrastarch
  • plasma protein fraction
  • hetastarch
  • rokitamycin
  • ridaforolimus
  • oleandomycin
  • patupilone
  • mitemcinal
  • midecamycin
  • mirvetuximab soravtansine
  • lorvotuzumab mertansine
  • kitasamycin
  • flurithromycin
  • eprinomectin
  • epofolate
  • epothilone D
  • coltuximab ravtansine
  • dirithromycin
  • doramectin
  • cethromycin
  • carbomycin
  • paramethasone
  • dexamethasone isonicotinate
  • quinupristin
  • sarilumab
  • dalfopristin
  • curcumin
  • luliconazole
  • procaine
  • chloroprocaine
  • phencyclidine
  • tenocyclidine
  • profenamine
  • halothane
  • lfenprodil
  • calcium levulinate
  • agmatine
  • calcium pangamate
  • calcium glubionate
  • edodekin alfa
  • beloranib
  • aflibercept
  • endostar
  • volociximab
  • roquinimex
  • anecortave acetate
  • squalamine
  • brolucizumab
  • trebananib
  • semaxanib
  • endostatin
  • halofuginone
  • resveratol
  • ranibizumab
  • fumagilin
  • bevacizumab
  • hyperforin
  • aminohippuric acid
  • opicapone
  • pafolacianine
  • bempedoic acid
  • belantamab mafodotin
  • prasterone
  • glecaprevir
  • levomenol
  • parachlorophenol
  • gadoxetic acid
  • cholecystokinin
  • caspofungin
  • ouabain
  • rifampicin
  • taurocholic acid
  • methylphosphinic acid
  • revefenacin
  • isoprenaline
  • posiphen
  • acotiamide
  • triflupromazine
  • pegvisomant
  • pipecuronium
  • regramostim
  • betaine
  • phenserine
  • diethylcarbamazine
  • cinchocaine
  • pancuronium
  • bambuterol
  • hexafluronium
  • aprotinin
  • tyrothricin
  • decamethonium
  • ipidacrine
  • tubocurarine
  • paraoxon
  • ginkgo biloba
  • methanesulfonyl fluoride
  • dichlorvos
  • fenthion
  • metrifonate
  • coumaphos
  • huperzine A
  • distigmine
  • neostigmine
  • isoflurophate
  • tasosartan
  • fimasartan
  • methylthioninium
  • minaprine
  • gallamine triethiodide
  • ambenonium
  • abiraterone
  • mibefradil
  • hydrocortisone (systemic)
  • cetirizine (systemic)
  • Talimogene Laherparepvec
  • Diacerein
  • Magnesium glucoheptonate
  • acyclovir and hydrocortisone
  • acyclovir (ophthalmic)
  • acyclovir (topical)
  • docosanol cream
  • camphor and phenol
  • dolutegravir, abacavir, and lamivudine
  • peramivir
  • lisdexamfetamine
  • ergoloid mesylates
  • memantine/donepezil
  • tranylcypromine
  • isocarboxazid
  • methenamine/sodium salicylate/benzoic acid
  • mometasone topical (Rx)
  • Esketamine intranasal
  • Oracit
  • Shohls Solution
  • sodium lactate
  • sodium citrate
  • lecanemab
  • donepezil (Rx)
  • donepezil transdermal
  • sodium thiosulfate
  • ciclopirox
  • undecylenic acid
  • butenafine
  • calcium and vitamin D
  • zoledronic acid
  • calcitonin salmon
  • pizotifen
  • indoramin
  • salicylic acid acne
  • minoxidil topical
  • adapalene
  • orlistat
  • COVID-19 subunit vaccine
  • amoxicillin /vonoprazan
  • levamlodipine (Rx)
  • Omeprazole, amoxicillin, and clarithromycin
  • simvastatin/ezetimibe
  • amlodipine/atorvastatin
  • amoxicillin and clavulanate potassium
  • lansoprazole, amoxicillin, and clarithromycin
  • noradrenaline
  • carbaryl
  • botulinum toxin
  • atropine
  • artemether/lumefantrine
  • ergonovine
  • bunazosin (Not available in the United States)
  • ibalizumab
  • dolutegravir
  • hydrocodone/pseudoephedrine
  • cetirizine/pseudoephedrine
  • acetaminophen/dextromethorphan/pseudoephedrine/guaifenesin
  • acetaminophen IV/ibuprofen IV (Pending FDA Approval)
  • medroxyprogesterone
  • acetaminophen/caffeine
  • Acetaminophen/magnesium salicylate/pamabrom
  • megestrol
  • pyridoxine (vitamin B6)
  • folic acid-cyanocobalamin-pyridoxine
  • L-methylfolate-pyridoxal 5′-phosphate-methylcobalamine
  • estropipate
  • betamethasone (systemic)
  • dolutegravir and lamivudine
  • zidovudine and lamivudine
  • mineral oil (oral/rectal)
  • regular insulin
  • dextromethorphan/bupropion
  • diphenhydramine/ibuprofen
  • enfuvirtide
  • doxapram
  • methamphetamine
  • dextroamphetamine
  • ephedrine
  • brompheniramine, dextromethorphan and phenylephrine
  • aspirin, chlorpheniramine, and phenylephrine
  • acetaminophen, pheniramine, and phenylephrine
  • chlorpheniramine and phenylephrine
  • guaifenesin and phenylephrine
  • rivastigmine
  • pyridostigmine
  • arecoline
  • physostigmine
  • abobotulinumtoxinA
  • echothiophate iodide
  • malathion
  • glibenclamide
  • rimabotulinumtoxinB
  • pioglitazone
  • daxibotulinumtoxinA
  • prabotulinumtoxinA
  • mepenzolate
  • trospium
  • modafinil
  • budesonide (oral inhalation)
  • budesonide (nasal)
  • budesonide (Topical)
  • vedolizumab
  • hydrocodone and homatropine
  • homatropine (ophthalmic)
  • methscopolamine
  • oxandrolone
  • nandrolone
  • fluoxymesterone
  • procyclidine
  • biperiden
  • benztropine
  • oxymetholone
  • ipratropium
  • belladonna/opium
  • pilocarpine
  • nicotine intranasal
  • succinylcholine
  • cromolyn sodium
  • mepolizumab
  • palivizumab
  • reslizumab
  • dupilumab
  • potassium iodide
  • benzralizumab
  • beclomethasone (nasal)
  • tetrahydrozoline
  • fluticasone (topical)
  • tecovirimat
  • entacapone
  • vaccinia immune globulin intravenous (Rx)
  • smallpox (vaccinia) vaccine, live
  • terazosin
  • labetalol 
  • smallpox and monkeypox vaccine (live, nonreplicating) (US: Availability limited to health department/CDC expanded access protocol) (Rx)
  • oxymetazoline
  • xylometazoline
  • meclizine
  • prazosin
  • belinostat
  • nabilone
  • tripelennamine
  • bismuth subcitrate, metronidazole and tetracycline
  • levalbuterol
  • rifaximin
  • cotrimoxazole
  • ethacrynic acid
  • senna
  • bisacodyl
  • sodium picosulfate, citric acid, and magnesium oxide
  • kaolin
  • anastrozole
  • docusate
  • cascara
  • dichlorphenamide
  • bismuth subsalicylate
  • methylcellulose
  • magnesium sulfate 
  • talazoparib
  • diphenoxylate/atropine
  • bacillus clausii
  • psyllium
  • bifidobacterium
  • lactobacillus
  • saccharomyces boulardii
  • lanreotide
  • cyproterone
  • ramucirumab (Rx)
  • fidaxomicin
  • tobramycin (systemic)
  • dacomitinib
  • pembrolizumab
  • amikacin (systemic)
  • panitumumab
  • blinatumomab
  • durvalumab
  • olaratumab
  • necitumumab
  • moxetumomab pasudotox
  • mogamulizumab
  • inotuzumab
  • dinutuximab
  • pentamycin
  • dibekacin
  • cemiplimab
  • gemtuzumab
  • demeclocycline
  • omadacycline
  • tobramycin (ophthalmic)
  • sarecycline
  • cefiderocol
  • valrubicin
  • plicamycin
  • denileukin diftitox
  • decitabine
  • niraparib
  • methacholine
  • carbachol
  • bethanechol
  • acetylcholine
  • atezolizumab
  • raloxifene
  • avelumab
  • leucovorin
  • cladabrine
  • pralatrexate
  • meclofenamate
  • pemetrexed
  • ustekinumab
  • diroximel fumarate
  • daratumumab
  • coccidioidin skin test
  • candida albicans extract
  • brewer’s yeast
  • poliovirus vaccine, live, trivalent
  • elotuzumab
  • trimetrexate
  • l-methyl folate
  • Methyclothiazide
  • Influenza virus vaccine
  • acitretin
  • tafamidis
  • sapropterin
  • Pidotimod
  • nitisinone
  • Mipomersen
  • levetiracetam
  • Inebilizumab
  • Diethylamine salicylate
  • COVID-19 vaccine
  • Cephalothin
  • alitretinoin
  • Alitretinoin
  • methotrexate
  • Verteporfin
  • Omacetaxine
  • methyl aminolevulinate topical
  • efgartigimod alfa
  • aminolevulinic acid
  • cetuximab
  • streptozocin
  • zoster vaccine recombinant
  • lyme disease vaccine
  • human papillomavirus vaccine
  • daclizumab
  • lomustiine
  • amitriptyline
  • triptorelin
  • Tedizolid
  • rituximab
  • darolutamide
  • Altretamine
  • Varicella-zoster vaccine
  • topotecan
  • ajmaline
  • pneumococcal vaccine
  • poliovirus vaccine
  • adenovirus vaccine type 7
  • adenovirus vaccine type 4
  • brincidofovir
  • lenograstim
  • ofatumumab
  • doxorubicin
  • thioguanine
  • tetanus toxoid
  • primidone
  • lipegfilgrastim
  • pegaspargase
  • monomethyl fumarate
  • ibritumomab
  • dimethyl fumarate
  • varicella-zoster vaccine (recombinant)
  • influenza virus vaccine, h5n1, live
  • carmustine
  • influenza virus vaccine (h5n1), adjuvanted
  • influenza a (h5n1) vaccine
  • eluxadoline
  • influenza virus vaccine quadrivalent, adjuvanted
  • idecabtagene vicleucel
  • adenovirus types 4 and 7 live, oral
  • thiotepa
  • tocilizumab
  • levodopa inhaled
  • efalizumab
  • canakinumab
  • aminoglutethimide
  • ado-trastuzumab emtansine
  • adenovirus vaccine
  • zoster vaccine live
  • typhoid vaccine, live
  • influenza virus vaccine, live, trivalent
  • influenza virus vaccine, h1n1, live
  • delavirdine
  • paclitaxel
  • siltuximab
  • miconazole
  • fludarabine
  • epirubicin
  • vinblastine
  • lomustine
  • risankizumab
  • rilonacept
  • pacritinib
  • linezolid
  • griseofulvin
  • vincristine
  • rufinamide
  • phenobarbital
  • nelarabine
  • mitoxantrone
  • mitomycin
  • mitapivat
  • letermovir
  • lasmiditan
  • idarubicin
  • filgrastim
  • elagolix
  • daunorubicin
  • daclatasvir
  • carfilzomib
  • brentuximab
  • anakinra
  • alefacept
  • thalidomide
  • teriflunomide
  • rubella virus vaccine
  • ozanimod
  • mumps virus vaccine
  • measles virus vaccine
  • golimumab
  • etanercept
  • certolizumab
  • adalimumab
  • etoposide
  • mechlorethamine
  • adenovirus type 7 vaccine
  • melphalan
  • palifermin
  • pimecrolimus
  • ropeginterferon alfa 2b
  • tacrolimus
  • tofacitinib
  • amphotericin B cholesteryl sulfate
  • amphotericin B deoxycholate
  • amphotericin B liposomal
  • amphotericin B phospholipid complex
  • anthrax vaccine adsorbed
  • denosumab
  • diphtheria & tetanus toxoids
  • echinacea
  • haemophilus influenzae type b vaccine
  • hepatitis A vaccine inactivated
  • hepatitis a/b vaccine
  • hepatitis b vaccine
  • HIV vaccine
  • human papillomavirus vaccine, quadrivalent
  • hydroxyurea
  • influenza virus vaccine (H5N1)
  • influenza virus vaccine trivalent
  • influenza virus vaccine trivalent, adjuvanted
  • influenza virus vaccine trivalent, recombinant
  • meningococcal A C Y and W-135 diphtheria conjugate vaccine
  • meningococcal A C Y and W-135 polysaccharide vaccine combined
  • meningococcal group B vaccine
  • ofatumumab SC
  • pneumococcal vaccine 13-valent
  • pneumococcal vaccine heptavalent
  • pneumococcal vaccine polyvalent
  • poliovirus vaccine inactivated
  • rabies vaccine
  • sipuleucel-T
  • trastuzumab
  • trastuzumab deruxtecan
  • eslicarbazepine acetate
  • vitamin A
  • rifampin
  • belzutifan
  • belimumab
  • belatacept
  • armodafinil
  • amobarbital
  • alemtuzumab
  • ocrelizumab
  • nivolumab
  • natalizumab
  • fingolimod
  • desogestrel
  • butalbital
  • brexanolone
  • zoster vaccine
  • yellow fever vaccine
  • varicella virus vaccine
  • smallpox vaccine
  • rotavirus vaccine
  • rubella vaccine
  • influenza virus vaccine quadrivalent
  • atracurium
  • dengue vaccine
  • tisagenlecleucel
  • lisocabtagene maraleucel
  • ciltacabtagene autoleucel
  • brexucabtagene autoleucel
  • axicabtagene ciloleucel
  • chlorambucil
  • ethinyl estradiol
  • dicumarol
  • atenolol
  • anisindione
  • penicillin G benzathine
  • sequelerin
  • chloramphenicol
  • heparin
  • enoxaparin
  • dalteparin
  • bivalirudin
  • argatroban
  • willow bark
  • bazedoxifene/conjugated estrogens
  • aspirin rectal
  • aspirin/citric acid/sodium bicarbonate
  • aspirin
  • ganaxolone
  • erythromycin stearate
  • erythromycin lactobionate
  • erythromycin ethylsuccinate
  • elbasvir/grazoprevir
  • daridorexant
  • cholera vaccine
  • lumacaftor/ivacaftor
  • dienogest/estradiol valerate
  • zafirlukast
  • urofollitropin
  • tralokinumab
  • torsemide
  • tazarotene
  • pseudoephedrine
  • propoxiphene napsylate
  • propoxiphene hydrochloride
  • oxyphencyclimine hydrochloride
  • oxymetazoline hydrochloride
  • naxitamab
  • nandrolone decanoate
  • methylphenidate
  • methocarbamol
  • idoxuridine
  • hyaluronidase
  • hyaluronic acid
  • gonadoreline hydrochloride
  • glycopyrrolate
  • ganirelix acetate
  • gallium citrate
  • fulvestrant
  • fexofenadine hydrochloride
  • fenefluramine hydrochloride
  • febuxostat
  • famciclovir
  • ergocalciferol
  • divalproex sodium
  • diclorfenamide
  • dezocine
  • desmopressin acetate
  • demeclocycline hydrochloride
  • defibrotide sodium
  • deferiprone
  • deferasirox
  • daunorubicin hydrochloride
  • darunavir
  • darifenacin hydrobromide
  • daptomycin
  • dapsone
  • dantrolene sodium
  • danazol
  • dalafampridine
  • dalbavancin Hydrochloride
  • daclatasvir dihydrochloride
  • dactinomycin
  • dacitabine
  • cefiderocol sulfate tosylate
  • butoconazole nitrate
  • benralizumab (Rx)
  • albuterol
  • acetylcysteine
  • acebutolol
  • acam2000
  • abrocitinib
  • abatacept
  • abametapir
  • abaloparatide
  • chloroquine
  • ferric maltol
  • lorlatinib
  • piracetam
  • timolol
  • chlorothiazide
  • ferric pyrophosphate citrate
  • lornoxicam
  • piretanide
  • tinidazole
  • chloroxylenol
  • ferric sulfate
  • lorpiprazole
  • pirfenidone
  • tiopronin
  • chlorpheniramine
  • ferrous bisglycinate
  • losartan
  • piroxicam
  • tiotropium
  • chlorpromazine
  • ferrous fumarate
  • lovastatin
  • pitavastatin
  • tipranavir
  • chlorpropamide
  • ferrous gluconate
  • loxoprofen
  • pitolisant
  • tirofiban
  • chlorprothixene
  • ferrous succinate
  • lubiprostone
  • pivampicillin
  • tisotumab vedotin
  • chlorthalidone
  • ferrous sulfate anhydrous
  • lumateperone
  • pivmecillinam
  • tixocortol
  • chlorzoxazone
  • ferumoxides
  • lumefantrine
  • plazomicin
  • tizanidine
  • abiraterone
  • cholecalciferolc
  • ferumoxsil
  • lumiracoxib
  • plerixafor
  • tobramycin (oral inhalation)
  • acalabrutinib
  • choline c 11
  • ferumoxytol
  • lurasidone
  • polatuzumab vedotin
  • tocainide
  • acarbose
  • choline magnesium trisalicylate
  • fesoterodine
  • lurbinectedin
  • polythiazide
  • tocofersolan
  • aceclofenac
  • choline salicylate
  • fexinidazole
  • lynestrenol
  • pomalidomide
  • tocopherol
  • acemetacin
  • chondroitin sulfate
  • finasteride
  • macimorelin
  • ponatinib
  • acenocoumarol
  • chromic chloride
  • finerenone (Rx)
  • macitentan
  • ponesimod
  • tolazamide
  • acetaminophen
  • chromic nitrate
  • fish oil
  • magaldrate
  • posaconazole
  • tolbutamide
  • acetazolamide
  • chromium
  • flavoxate
  • magnesium
  • potassium
  • tolcapone
  • acetohexamide
  • chromium gluconate
  • flecainide
  • magnesium carbonate
  • potassium acetate
  • tolfenamic acid
  • acetylsalicylic acid
  • chromium nicotinate
  • flibanserin
  • magnesium chloride
  • potassium bicarbonate
  • tolmetin
  • acipimox
  • chromous sulfate
  • floctafenine
  • magnesium citrate
  • potassium cation
  • tolterodine
  • aclidinium
  • ciclesonide
  • florbetaben (18f)
  • magnesium gluconate
  • potassium chloride
  • tolvaptan
  • acrivastine
  • cidofovir
  • florbetapir (18f)
  • magnesium hydroxide
  • potassium citrate
  • topiramate
  • acyclovir
  • cilazapril
  • floxuridine
  • magnesium oxide
  • potassium nitrate
  • adefovir dipivoxil
  • cilostazol
  • flucloxacillin
  • magnesium silicate
  • potassium perchlorate
  • torasemide
  • adenosine
  • cimetidine
  • fluconazole
  • potassium sulfate
  • toremifene
  • agomelatine
  • cinacalcet
  • flucytosine
  • magnesium trisilicate
  • tositumomab
  • albendazole
  • cinnarizine
  • fludeoxyglucose (18f)
  • mangafodipir
  • pralidoxime
  • trabectedin
  • albiglutide
  • cinoxacin
  • fludrocortisone
  • manidipine
  • pralsetinib
  • tramadol
  • albutrepenonacog alfa
  • ciprofibrate
  • fluindione
  • mannitol
  • pramipexole
  • trametinib
  • alclofenac
  • cisapride
  • flumazenil
  • maprotiline
  • pramlintide
  • trandolapril
  • aldesleukin
  • cisplatin
  • flumethasone
  • maraviroc
  • prasugrel
  • trastuzumab emtansine
  • alectinib
  • citalopram
  • flunarizine
  • maribavir
  • pravastatin
  • trazodone
  • alendronic acid
  • cladribine
  • flunisolide
  • mebeverine
  • prazepamb
  • treprostinil
  • alfentanil
  • clarithromycin
  • flunitrazepam
  • mecamylamine
  • praziquantel
  • tretinoin
  • alfuzosin
  • clemastine
  • fluocinolone acetonide
  • mecasermin
  • prednisolone
  • triamcinolone
  • alimemazine
  • clevidipine
  • fluocinonide
  • meclofenamic acid
  • prednisolone acetate
  • triamterene
  • aliskiren
  • clindamycin
  • fluocortolone
  • medrogestone
  • prednisolone phosphate
  • triazolam
  • allopurinol
  • clobazam
  • fluorouracil
  • medroxyprogesterone acetate
  • prednisone (Rx)
  • trichlormethiazide
  • almasilate
  • clobetasol propionate
  • fluoxetine
  • mefenamic acid
  • prednisone acetate
  • triclabendazole
  • almotriptan
  • clofarabine
  • flupentixol
  • mefloquine
  • pregabalin
  • triethylenetetramine
  • alogliptin
  • clofazimine
  • fluprednisolone
  • megestrol acetate
  • pregnenolone
  • trifluoperazine
  • alosetron
  • clofibrate
  • flurazepam
  • melatonin
  • prenylamine
  • trifluridine
  • alpelisib
  • clomipramine
  • flurbiprofen
  • meloxicam
  • pretomanid
  • trilaciclib
  • alprazolam
  • fluspirilene
  • memantine
  • primaquine
  • trilostane
  • clonidine
  • flutamide
  • menthyl salicylate
  • probenecid
  • trimebutine
  • aluminium phosphate
  • clopidogrel
  • fluticasone (nasal)
  • meperidine
  • probucol
  • trimethadione
  • aluminum hydroxide
  • clorazepic acid
  • fluticasone furoate
  • mephenytoin
  • procainamide
  • trimethoprim
  • amantadine
  • clotiazepam
  • fluticasone propionate
  • mepivacaine
  • procaine benzylpenicillin
  • ambrisentan (Rx)
  • clove oil
  • fluvastatin
  • meprednisone
  • procarbazine
  • trimipramine
  • ambroxol
  • cloxacillin
  • fluvoxamine
  • mepyramine
  • prochlorperazine
  • triprolidine
  • amifampridine
  • folic acid
  • mercaptopurine
  • progesterone
  • amikacin (oral inhalation)
  • fomepizole
  • meropenem
  • promazine
  • troglitazone
  • amiloride
  • fondaparinux
  • mesalazine
  • promethazine
  • troleandomycin
  • aminophenazone
  • clonazepam
  • formestane
  • mesoridazine
  • propafenone
  • tropisetron
  • aminophylline
  • formoterol
  • mestranol
  • propantheline
  • trovafloxacin
  • amiodarone
  • fosamprenavir
  • metamfetamine
  • propiverine
  • tucatinib
  • amisulpride
  • fosaprepitant
  • metamizole
  • propofol
  • typhoid vaccine
  • foscarnet
  • metaxalone
  • propranolol
  • ubidecarenone
  • amlodipine
  • fosfomycin
  • metformin
  • propylthiouracil
  • ubrogepant
  • ammonium chloride
  • fosinopril
  • methadone
  • protriptyline
  • udenafil
  • amodiaquine
  • clozapine
  • fosnetupitant
  • methazolamide
  • prucalopride
  • ulipristal
  • amoxapine
  • cobicistat
  • fosphenytoin
  • methimazole
  • prussian blue
  • upadacitinib
  • amoxicillin
  • cobimetinib
  • fostamatinib
  • pyrantel
  • vaborbactam
  • amphetamine
  • cocaine
  • fostemsavir
  • methotrimeprazine
  • pyrazinamide
  • valaciclovir
  • amphotericin b
  • codeine
  • framycetin
  • methoxsalen
  • valbenazine
  • ampicillin
  • colchicine
  • frovatriptan
  • methsuximide
  • pyrimethamine
  • valdecoxib
  • amprenavir
  • colistimethate
  • furosemide
  • methyldopa
  • pyrithione
  • valganciclovir
  • amrinone
  • colistin
  • fusidic acid
  • methylene blue
  • quazepam
  • valproic acid
  • anagrelide
  • conivaptan
  • gabapentin enacarbil
  • methylergometrine
  • quetiapine
  • valsartan
  • ancestim
  • conjugated estrogens
  • gadobenic acid
  • methylnaltrexone
  • vancomycin
  • antazoline
  • copanlisib
  • gadodiamide
  • methylprednisolone
  • quinapril
  • vandetanib
  • corifollitropin alfa
  • gadofosveset trisodium
  • methylprednisolone aceponate
  • quinethazone
  • vardenafil
  • corticotropin
  • gadopentetic acid
  • methylprednisolone hemisuccinate
  • quinidine
  • varenicline
  • cortisone acetate
  • gadoteric acid
  • methylprednisone
  • quinine
  • velpatasvir
  • antrafenine
  • crizotinib
  • gadoteridol
  • methyltestosterone
  • rabeprazole
  • vemurafenib
  • apalutamide
  • cyanocobalamin
  • galantamine
  • methysergide
  • raltegravir
  • venetoclax
  • apixaban
  • cyclacillin
  • ganciclovir
  • meticillin
  • ramelteon
  • venlafaxine
  • apomorphine
  • cyclandelate
  • gatifloxacin
  • meticrane
  • ramipril
  • verapamil
  • apremilast
  • cyclizine
  • gefitinib
  • metoclopramide
  • ranitidine
  • vernakalant
  • aprepitant
  • cyclobenzaprine
  • gemcitabine
  • metolazone
  • ranolazine
  • vibrio cholerae cvd 103-hgr strain live antigen
  • arformoterol
  • cyclopenthiazide
  • gemfibrozil
  • metoprolol
  • rasagiline
  • vilanterol
  • aripiprazole
  • cyclophosphamide
  • gemifloxacin
  • metronidazole
  • reboxetine
  • vilazodone
  • aripiprazole lauroxil
  • cyclosporine
  • gentamicin
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  • arsenic trioxide
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  • mifepristone
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  • atazanavir
  • dapagliflozin
  • glimepiride
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  • vitamin d
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  • ribavirin
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  • glyburide
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  • minocycline
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  • guanfacine
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  • azelastine
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  • moxifloxacin
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  • haloperidol
  • muzolimine
  • ritonavir
  • zinc
  • azlocillin
  • dexlansoprazole
  • hetacillin
  • mycophenolate mofetil
  • rivaroxaban
  • zinc acetate
  • aztreonam
  • dexmedetomidine
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  • mycophenolic acid
  • rizatriptan
  • zinc ascorbate
  • bacampicillin
  • dexpanthenol
  • hydralazine
  • n-acetyltyrosine
  • rofecoxib
  • zinc chloride
  • bacitracin
  • dexrazoxane
  • hydrochlorothiazide
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  • zinc gluconate
  • baclofen
  • dextran
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  • dichlorobenzyl alcohol
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  • naloxegol
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  • bendamustine
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  • hydromorphone
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  • bendroflumethiazide
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  • hydrotalcite
  • naproxen
  • rucaparib
  • zotepine
  • dicyclomine
  • hydroxocobalamin
  • nateglinide
  • rupatadine
  • zuclopenthixol
  • benoxaprofen
  • didanosine
  • hydroxychloroquine
dicyclomine + 

glucagon

it increases the toxicity of dicyclomine

glucagon intranasal

it increases the toxicity of dicyclomine

pramlintide

pramlintide and dicyclomine increase the effect of each other through a synergistic activity

revefenacin

dicyclomine decreases the effect of revefenacin by decreasing the cholinergic transmission

secretin

dicyclomine decreases the effect of secretin by antagonistic activity

umeclidinium bromide

umeclidinium bromide and dicyclomine increase the toxicity of each other by synergism

ramosetron

anticholinergic agents increase the constipating activity of ramosetron

mianserin

it increases the anticholinergic agents

dimenhydrinate

dimenhydrinate increases the toxicity of dicyclomine due to pharmacodynamic synergism

donepezil

it decreases the effect of dicyclomine by antagonistic activity

galantamine

it decreases the effect of dicyclomine by antagonistic activity

trazodone

trazodone and dicyclomine decrease the cholinergic transmission

 

Dosage forms & Strengths 

Capsule 

10 mg 

Tablet 

20 mg 

Injectable solution 

10mg/ml 

Syrup 

10mg/5ml 

Irritable Bowel Syndrome 

20 mg of dicyclomine is indicated orally every 6 hours
The dose can be increased to 40 mg every 6 hours if efficacy is not attained within 2 weeks
The maximum dose in the case of irritable bowel syndrome is 80 mg per day
For injection dose, 10-20 mg of the intramuscular dose every 6 hours is optimum
Dose consideration
The intramuscular dose should not be used for more than 1-2 days
Replace it with an oral dose as soon as possible
Do not use intravenous dose



 

Dosage forms & Strengths 

Capsule 

10 mg 

Tablet 

20 mg 

Injectable solution 

10mg/ml 

Syrup 

10mg/5ml 

Irritable Bowel Syndrome (IBS) 

For infants of > 6 months of age: 5 mg orally every 6 to 8 hours
Do not exceed the dose of more than 20mg/day
Children: 10 mg orally every 6 to 8 hours
The dose should not exceed 40mg orally per day



 

Dosage forms & Strengths 

Capsule 

10 mg 

Tablet 

20 mg 

Injectable solution 

10mg/ml 

Syrup 

10mg/5ml 

Irritable Bowel Syndrome (IBS) 

10-20 mg of the oral dose every 6 hours is recommended for geriatrics
Do not exceed the dose of more than 160 mg/day
Intramuscular injections are not advised for geriatric patients



Frequency defined 

>10% 

Dry mouth  

Dizziness  

Blurred vision 

1-10% 

Nervousness 

Weakness 

Somnolence 

Frequency not defined 

Abdominal distension 

Confusion state 

Cycloplegia 

Delirium 

Dermatitis 

Erythema 

Fatigue 

Hallucinations 

Insomnia 

Malaise 

Palpitation 

Rash 

Syncope 

Contraindication/Caution: 

dicyclomine has several contraindications and precautions that should be considered before use. These include: 

  • Hypersensitivity: dicyclomine should not be used in patients who have a known hypersensitivity to the medication or any of its components. 
  • Glaucoma: dicyclomine should be used with caution in patients with narrow-angle glaucoma, as it can increase intraocular pressure and exacerbate the condition. 
  • Gastrointestinal obstruction: dicyclomine should not be used in patients with obstructive disorders of the GI tract, such as pyloric stenosis or paralytic ileus. 
  • Severe ulcerative colitis: dicyclomine should be used with caution in patients with severe ulcerative colitis, as it may lead to toxic megacolon. 
  • Myasthenia gravis: dicyclomine should be used with caution in patients with myasthenia gravis, as it can exacerbate muscle weakness. 
  • Children: dicyclomine should not be used in children under 6 months of age, as it can cause serious side effects. 
  • Pregnancy and breastfeeding: dicyclomine should only be used during pregnancy or breastfeeding if the potential benefits outweigh the potential risks. 

Overall, dicyclomine should be used with caution in patients with certain medical conditions and should only be used under the guidance of a healthcare professional. It is important to inform the healthcare provider of any pre-existing medical conditions or medications being taken before starting dicyclomine therapy. 

Pregnancy consideration:  

Category B 

Breastfeeding warnings: dicyclomine should not be taken by lactating females 

Pregnancy category: 

  • Category A: Satisfactory and well-controlled studies show no risk to the fetus in the first or later trimester. 
  • Category B: There is no affirmation of risk to the fetus found in animal reproduction studies, and there are not enough studies on pregnant women. 
  • Category C: Adverse effects on the fetus found with evidence in animal reproduction studies and no adequate evidence for a product in humans; Pregnant women must take care of the potential risks. 
  • Category D: There is adequate data available with sufficient evidence of human fetal risk from various platforms. However, despite potential dangers may be used only in emergency cases for potential benefits. 
  • Category X: Drugs listed in this category outweigh the risks over benefits. The drug is not for pregnant women. 
  • Category N: No data is available for the drug under this category. 

Pharmacology: 

dicyclomine is a medication that belongs to the class of anticholinergic drugs, and it works by blocking the action of acetylcholine at muscarinic receptors in the smooth muscles of the gastrointestinal (GI) tract. This leads to relaxation of the smooth muscles and a decrease in spasms, which can help to reduce abdominal pain and cramping associated with various GI disorders. 

dicyclomine is rapidly absorbed after oral administration, and it reaches peak plasma concentrations within 1 to 1.5 hours. The medication is metabolized in the liver and excreted in the urine and feces. The half-life of dicyclomine is approximately 1.5 to 2 hours, and the duration of action is 4 to 6 hours. 

In addition to its antispasmodic effects, dicyclomine also has some local anesthetic effects on the GI tract, which can help to reduce pain and discomfort associated with GI spasms. dicyclomine can also reduce the secretion of gastric acid, which can be helpful in the treatment of peptic ulcers. 

Pharmacodynamics: 

dicyclomine is an anticholinergic medication that works by blocking the action of acetylcholine at muscarinic receptors in the smooth muscles of the gastrointestinal (GI) tract. This leads to the relaxation of the smooth muscles and a decrease in spasms, which can help to reduce abdominal pain and cramping associated with various GI disorders. 

Acetylcholine is a neurotransmitter that stimulates smooth muscle contraction in the GI tract, and its effects are mediated through muscarinic receptors. dicyclomine competitively inhibits the binding of acetylcholine to muscarinic receptors, leading to reduced smooth muscle contractions and an overall decrease in GI spasms. 

In addition to its antispasmodic effects, dicyclomine also has some local anesthetic effects on the GI tract, which can help to reduce pain and discomfort associated with GI spasms. dicyclomine can also reduce the secretion of gastric acid, which can be helpful in the treatment of peptic ulcers. 

Pharmacokinetics: 

Absorption 

The bioavailability is 67% in an intramuscular injection 

The onset of action is 1-2 hours 

The duration of action is 4 hours 

The peak plasma concentration for oral is achieved in 60-90 min 

Distribution 

The volume of distribution is 3.65 L/kg 

Metabolism 

The drug gets extensively metabolized in the liver 

Elimination and Excretion 

The half-life is 1.8 hours 

The drug is excreted 80% in urine and 8% in feces

Administration: 

dicyclomine is usually taken orally, and it is available in the form of capsules, tablets, or an oral solution. The medication should be taken with water, and it can be taken with or without food. 

The dosage and frequency of dicyclomine administration depend on the specific condition being treated and the patient’s age, weight, and overall health. Typically, the recommended adult dose of dicyclomine for the treatment of functional bowel/irritable bowel syndrome is 20 mg four times daily, with the maximum dose of 40 mg four times daily. 

For children, the recommended dose of dicyclomine is based on weight and is usually lower than the adult dose. The medication should not be used in children under six months of age. 

dicyclomine should be taken as prescribed by a healthcare professional, and patients should not exceed the recommended dose or frequency of administration. It is important to follow the instructions provided by the healthcare professional and to continue taking the medication for the entire duration of the prescribed treatment. 

Patient information leaflet 

Generic Name: dicyclomine 

Pronounced: dye-SYE-kloe-meen 

Why do we use dicyclomine? 

dicyclomine is a medication that is used to treat various gastrointestinal (GI) conditions that involve spasms, cramps, and pain. It is primarily used to treat functional bowel/irritable bowel syndrome, that is characterized by abdominal pain and discomfort, bloating, and changes in bowel habits. 

In addition to functional bowel/irritable bowel syndrome, dicyclomine can also be used to treat other GI conditions, including: 

  • Gastric ulcers 
  • Gastroesophageal reflux disease (GERD) 
  • Intestinal hypermotility 
  • Colitis 
  • Pancreatitis 
  • Diverticulitis 

dicyclomine works by relaxing the smooth muscles in the GI tract, which can help to reduce spasms and pain associated with these conditions. It can also reduce the secretion of gastric acid, which can be helpful in the treatment of peptic ulcers. 

Overall, dicyclomine is a medication that acts on the smooth muscles of the GI tract to reduce spasms and pain associated with various GI disorders. It is important to note that dicyclomine is a prescription medication and should only be used under the guidance of a healthcare professional. 

ADVERTISEMENT 

dicyclomine

Brand Name :

Bentyl

Synonyms :

dicyclomine

Class :

Anticholinergic agents




No data available for drug.

Dosage forms & Strengths 

Capsule 

10 mg 

Tablet 

20 mg 

Injectable solution 

10mg/ml 

Syrup 

10mg/5ml 

irritable Bowel Syndrome 

20 mg of dicyclomine is indicated orally every 6 hours
The dose can be increased to 40 mg every 6 hours if efficacy is not attained within 2 weeks
The maximum dose in the case of irritable bowel syndrome is 80 mg per day
For injection dose, 10-20 mg of the intramuscular dose every 6 hours is optimum
Dose consideration
The intramuscular dose should not be used for more than 1-2 days
Replace it with an oral dose as soon as possible
Do not use intravenous dose



Dosage forms & Strengths 

Capsule 

10 mg 

Tablet 

20 mg 

Injectable solution 

10mg/ml 

Syrup 

10mg/5ml 

irritable bowel syndrome (IBS) 

For infants of > 6 months of age: 5 mg orally every 6 to 8 hours
Do not exceed the dose of more than 20mg/day
Children: 10 mg orally every 6 to 8 hours
The dose should not exceed 40mg orally per day



Dosage forms & Strengths 

Capsule 

10 mg 

Tablet 

20 mg 

Injectable solution 

10mg/ml 

Syrup 

10mg/5ml 

irritable bowel syndrome (IBS) 

10-20 mg of the oral dose every 6 hours is recommended for geriatrics
Do not exceed the dose of more than 160 mg/day
Intramuscular injections are not advised for geriatric patients



DRUG INTERACTION

dicyclomine

&

  • prednisolone and gentamicin ophthalmic
  • promethazine and codeine
  • poractant alfa
  • protamine sulfate
  • aflibercept intravitreal
  • prednicarbate
  • promethazine/dextromethorphan
  • codeine, phenylephrine, and promethazine
  • potassium phosphate
  • glatiramer acetate
  • gentamicin (Ophthalmic)
  • leniolisib
  • rezafungin
  • fluorometholone
  • dalfampridine
  • hydrocortisone topical 
  • empagliflozin and linagliptin
  • triamcinolone topical
  • minocycline topical
  • minocycline dental
  • ketotifen ophthalmic
  • darunavir and cobicistat
  • lidocaine topical
  • neomycin/polymyxin B/bacitracin/lidocaine (OTC)
  • lidocaine/ hydrocortisone
  • lidocaine anesthetic
  • lidocaine ophthalmic
  • lidocaine/tetracaine
  • desonide
  • dabigatran
  • fexofenadine
  • fluoride
  • decitabine and cedazuridine
  • dasiglucagon
  • hydroxypropyl cellulose ophthalmic
  • epoetin alfa
  • ibritumomab tiuxetan
  • trimethobenzamide
  • dexamethasone/ tobramycin
  • tafasitamab
  • valacyclovir
  • mebendazole
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  • flaxseed
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  • horseradish
  • ziv-aflibercept
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  • tildrakizumab
  • sulopenem (Pending FDA Approval)
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  • birch
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  • tafluprost
  • methohexital
  • urea and hydrocortisone
  • unoprostone ophthalmic
  • trihexyphenidyl
  • ezetimibe
  • evolocumab
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  • methenamine
  • misoprostol
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  • valerian
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  • hydrocortisone acetic acid otic
  • butorphanol
  • butoconazole
  • adapalene and benzoyl peroxide
  • acrivastine and pseudoephedrine
  • neomycin/polymyxin B/bacitracin topical
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  • econazole topical
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  • aspirin/dipyridamole
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  • difenoxin and atropine
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  • allogeneic cultured keratinocytes/fibroblasts in bovine collagen
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  • cyclopentolate
  • polymyxin B/bacitracin topical
  • ketoconazole topical
  • tavaborole
  • tagraxofusp
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  • sacubitril/valsartan
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  • dextrose
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  • iohexol
  • ferric citrate
  • elapegademase
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  • danaparoid
  • dantrolene
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  • edaravone
  • amcinonide
  • carglumic acid
  • alcaftadine ophthalmic
  • agalsidase beta
  • afamelanotide
  • fosdenopterin
  • lidocaine and chlorhexidine
  • levorphanol
  • calcifediol
  • factor VIIa, recombinant
  • triheptanoin
  • peanut oral allergen powder
  • teprotumumab
  • poly-L-lactic acid/carboxymethylcellulose/mannitol
  • xenon Xe 129 hyperpolarized
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  • glatiramer
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  • cycloserine
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  • nadofaragene firadenovec
  • ozenoxacin
  • guaifenesin
  • adagrasib
  • guselkumab
  • adalimumab-aacf
  • nonoxynol-9
  • nifurtimox
  • nusinersen
  • nitazoxanide
  • mavacamten
  • calcipotriene
  • bimatoprost
  • obinutuzumab
  • amifostine
  • oxycodone/​aspirin
  • oxycodone/ibuprofen
  • oteseconazole
  • oxychlorosene
  • porfimer
  • pramoxine /hydrocortisone topical
  • podofilox
  • quinapril/hydrochlorothiazide
  • acetaminophen/pamabrom/pyrilamine
  • levobunolol
  • paregoric
  • idursulfase
  • lesinurad and allopurinol
  • latanoprost/​netarsudil ophthalmic
  • lactase enzyme
  • bioadherent oral
  • latanoprost and timolol
  • latanoprostene bunod
  • ledipasvir/sofosbuvir
  • imipenem/cilastatin/relebactam
  • imipenem/cilastatin
  • hemin
  • deucravacitinib
  • house dust mite allergen extract
  • halobetasol topical/tazarotene
  • remimazolam
  • somatropin
  • remifentanil
  • ethotoin
  • etidronate
  • empagliflozin, linagliptin, and metformin
  • elvitegravir/cobicistat/emtricitabine/tenofovir AF
  • empagliflozin/​linagliptin
  • evinacumab
  • finasteride and tadalafil
  • flortaucipir (18F)
  • proparacaine/ fluorescein ophthalmic
  • fluorescein/benoxinate ophthalmic
  • fluphenazine
  • alogliptin/​metformin
  • alogliptin/pioglitazone
  • alitretinoin topical
  • dextrose/ sodium citrate/fructose
  • dasabuvir
  • ombitasvir​/paritaprevir/​ritonavir
  • hydrocodone/​chlorpheniramine/​pseudoephedrine
  • hydroxyamphetamine/​tropicamide
  • acamprosate
  • gadobutrol
  • teclistamab
  • tremelimumab
  • futibatinib
  • etranacogene dezaparvovec
  • olutasidenib
  • naproxen and diphenhydramine
  • naratriptan
  • gadopiclenol
  • gadoxetate
  • gadoversetamide
  • naphazoline/pheniramine
  • naphazoline
  • nalbuphine
  • vosoritide
  • vitamin K1 (phytonadione)
  • moxidectin
  • basiliximab
  • fecal microbiota, live-jslm
  • ibuprofen/famotidine
  • famotidine
  • raxibacumab
  • omalizumab
  • measles, mumps, rubella, and varicella vaccine, live (Rx)
  • senna/docusate
  • dinoprostone
  • measles mumps and rubella vaccine, live
  • immune globulin IM (IGIM)
  • dyclonine
  • doravirine, lamivudine, and tenofovir disoproxil fumarate
  • elexacaftor/tezacaftor/ivacaftor
  • ivacaftor/tezacaftor
  • treosulfan
  • tranexamic acid
  • norethindrone acetate/​estradiol/​elagolix
  • artesunate
  • trientine
  • trifarotene
  • ziconotide
  • vonoprazan/amoxicillin/clarithromycin
  • pyrithione zinc
  • zinc oxide topical
  • naphazoline/​zinc sulfate/​glycerin ophthalmic
  • voretigene neparvovec
  • nirmatrelvir/ritonavir
  • bebetelovimab
  • sodium chloride
  • relugolix/​estradiol/​norethindrone
  • defibrotide
  • prothionamide
  • liraglutide
  • maitake
  • etilfrine
  • alpha-lipoic acid
  • ramosetron
  • olodaterol/tritropium
  • cimetropium
  • umeclidinium
  • itopride
  • secretin
  • naftopidil
  • trimeprazine
  • benperidol
  • chlormethiazole
  • multivitamins
  • secukinumab
  • glycopyrrolate inhaled and formoterol
  • amitriptyline and chlordiazepoxide
  • tirzepatide
  • relugolix/estradiol/norethindrone
  • mupirocin
  • alvimopan
  • chlordiazepoxide
  • insulin regular human
  • insulin aspart protamine/​insulin aspart
  • insulin isophane human/​insulin regular human
  • insulin degludec/insulin aspart
  • teplizumab
  • chlordiazepoxide/clidinium
  • aspirin, sodium bicarbonate, and citric acid
  • aluminum hydroxide, magnesium hydroxide, and simethicone
  • glycopyrrolate inhaled
  • olodaterol/tiotropium
  • umeclidinium bromide
  • timolol/dorzolamide
  • travoprost ophthalmic
  • loxapine
  • eptifibatide
  • hydrocodone/acetaminophen
  • omega 3 fatty acids
  • trandolapril/​verapamil
  • abciximab
  • artificial saliva
  • diphtheria, hepatitis B, pertussis (acellular), polio, and tetanus vaccine
  • diphtheria, haemophilus B, pertussis, polio, tetanus vaccine
  • haemophilus influenzae type b vaccine/hepatitis b vaccine
  • butalbital/aspirin/caffeine 
  • colchicine/probenecid
  • atovaquone and proguanil
  • ursodiol
  • chenodiol
  • casirivimab/imdevimab
  • tixagevimab/cilgavimab
  • molnupiravir
  • bebtelovimab
  • calcium, magnesium, potassium and sodium oxybate
  • sodium oxybate
  • diphtheria, polio, pertussis acellular, tetanus vaccine
  • pseudoephedrine loratadine
  • sodium chloride nasal
  • hydroxychloroquine sulfate
  • atorvastatin and ezetimibe
  • teriparatide
  • alendronate and cholecalciferol
  • alprostadil (IV)
  • romosozumab
  • risedronate
  • alendronate
  • glyburide/metformin
  • clorazepate
  • rosuvastatin/​ezetimibe
  • paclitaxel/encequidar
  • valsartan/amlodipine
  • enalapril/hydrochlorothiazide
  • enalapril and felodipine
  • amiloride/hydrochlorothiazide
  • triamterene/hydrochlorothiazide
  • lisinopril/hydrochlorothiazide
  • tegaserod
  • rhein
  • ritanserin
  • sulfaphenazole
  • sulconazole
  • taurursodiol
  • bromeperidol
  • carbapenems
  • fotemustine
  • difelikefalin
  • bromopride
  • alizapride
  • olopatadine
  • oxomemazine
  • paraldehyde
  • oxcarbazepine
  • kratom
  • elexacaftor
  • oritavancin
  • miocamycin
  • curcumin sulfate
  • seproxetine
  • clotrimazole
  • remacemide
  • piperine
  • ditiocarb
  • danoprevir
  • oxetacaine
  • topiroxostat
  • indisulam
  • tofisopam
  • noscapine
  • thiopental
  • tioconazole
  • nicotinamide
  • rutin
  • mequitazine
  • somatostatin
  • vapreotide
  • econazole
  • saracatinib
  • lestaurtinib
  • efonidipine
  • zimelidine
  • indalpine
  • desvenlafaxine
  • benidipine
  • dapoxetine
  • tesmilifene
  • pergolide
  • sitaxentan
  • resveratrol
  • bifonazole
  • tildipirosin
  • solithromycin
  • selamectin
  • imiquimod topical
  • fluorouracil topical
  • peginterferon alfa-2b
  • interferon alfa-2b
  • alteplase
  • tanshinone I
  • rosmarinic acid
  • caryophyllene
  • ursolic acid
  • cepharanthine
  • veliflapon
  • mirikizumab
  • cp-96345
  • famprofazone
  • peoniflorin
  • fepradinol
  • licofelone
  • polmacoxib
  • ebselen
  • taxifolin
  • betulinic acid
  • flurbiprofen axetil
  • talniflumate
  • morniflumate
  • nitroaspirin
  • firocoxib
  • ns-398
  • cimicoxib
  • robenacoxib
  • sc-236
  • imidazole salicylate
  • trolamine salicylate
  • pirprofen
  • benorilate
  • ethenzamide
  • mofebutazone
  • proquazone
  • carbaspirin calcium
  • guacetisal
  • proglumetacin
  • propyphenazone
  • pranoprofen
  • bendazac
  • tenidap
  • lonazolac
  • nifenazone
  • flunoxaprofen
  • difenpiramide
  • feprazone
  • bufexamac
  • alminoprofen
  • suxibuzone
  • fentiazac
  • tinoridine
  • tepoxalin
  • indobufen
  • flunixin
  • propacetamol
  • clonixin
  • droxicam
  • epirizole
  • etofenamate
  • ibuproxam
  • indoprofen
  • kebuzone
  • felbinac
  • zaltoprofen
  • azapropazone
  • zomepirac
  • niflumic acid
  • magnesium salicylate
  • suprofen
  • nepafenac
  • bromfenac
  • ciprofloxacin and hydrocortisone (otic) (Rx)
  • hydrocortisone/neomycin/polymyxin otic (Rx)
  • vigabatrine
  • valproate
  • tezepelumab (Rx)
  • triamcinolone acetonide/nystatin
  • triamcinolone suprachoroidal (Rx)
  • triamcinolone, intranasal
  • ciclesonide inhaled
  • diosmin
  • tirbanibulin
  • padeliporfin
  • roxadustat
  • aminosalicylic acid
  • rasburicase
  • tetracaine
  • articaine
  • ropivacaine
  • nitrous oxide
  • sulfapyridine
  • sulfanilamide
  • mafenide
  • isometheptene
  • amyl nitrite
  • antipyrine
  • isosorbide dinitrate
  • prilocaine
  • nitroglycerin
  • tobacco
  • batefenterol
  • hexoprenaline
  • pf-00610355
  • racepinephrine
  • protokylol
  • doxofylline
  • phenylpropanolamine
  • isoetharine
  • ephedra sinica root
  • dipivefrin
  • arbutamine
  • norepinephrine
  • fenoterol
  • clenbuterol
  • pirbuterol
  • epinephrine
  • ritodrine
  • procaterol
  • orciprenaline
  • bitolterol
  • abediterol
  • fluticasone furoate, umeclidinium and vilanterol
  • fluticasone furoate and vilanterol
  • mometasone and formoterol
  • pramoxine topical (OTC)
  • menthol/pramoxine (topical)
  • tetrastarch
  • plasma protein fraction
  • hetastarch
  • rokitamycin
  • ridaforolimus
  • oleandomycin
  • patupilone
  • mitemcinal
  • midecamycin
  • mirvetuximab soravtansine
  • lorvotuzumab mertansine
  • kitasamycin
  • flurithromycin
  • eprinomectin
  • epofolate
  • epothilone D
  • coltuximab ravtansine
  • dirithromycin
  • doramectin
  • cethromycin
  • carbomycin
  • paramethasone
  • dexamethasone isonicotinate
  • quinupristin
  • sarilumab
  • dalfopristin
  • curcumin
  • luliconazole
  • procaine
  • chloroprocaine
  • phencyclidine
  • tenocyclidine
  • profenamine
  • halothane
  • lfenprodil
  • calcium levulinate
  • agmatine
  • calcium pangamate
  • calcium glubionate
  • edodekin alfa
  • beloranib
  • aflibercept
  • endostar
  • volociximab
  • roquinimex
  • anecortave acetate
  • squalamine
  • brolucizumab
  • trebananib
  • semaxanib
  • endostatin
  • halofuginone
  • resveratol
  • ranibizumab
  • fumagilin
  • bevacizumab
  • hyperforin
  • aminohippuric acid
  • opicapone
  • pafolacianine
  • bempedoic acid
  • belantamab mafodotin
  • prasterone
  • glecaprevir
  • levomenol
  • parachlorophenol
  • gadoxetic acid
  • cholecystokinin
  • caspofungin
  • ouabain
  • rifampicin
  • taurocholic acid
  • methylphosphinic acid
  • revefenacin
  • isoprenaline
  • posiphen
  • acotiamide
  • triflupromazine
  • pegvisomant
  • pipecuronium
  • regramostim
  • betaine
  • phenserine
  • diethylcarbamazine
  • cinchocaine
  • pancuronium
  • bambuterol
  • hexafluronium
  • aprotinin
  • tyrothricin
  • decamethonium
  • ipidacrine
  • tubocurarine
  • paraoxon
  • ginkgo biloba
  • methanesulfonyl fluoride
  • dichlorvos
  • fenthion
  • metrifonate
  • coumaphos
  • huperzine A
  • distigmine
  • neostigmine
  • isoflurophate
  • tasosartan
  • fimasartan
  • methylthioninium
  • minaprine
  • gallamine triethiodide
  • ambenonium
  • abiraterone
  • mibefradil
  • hydrocortisone (systemic)
  • cetirizine (systemic)
  • Talimogene Laherparepvec
  • Diacerein
  • Magnesium glucoheptonate
  • acyclovir and hydrocortisone
  • acyclovir (ophthalmic)
  • acyclovir (topical)
  • docosanol cream
  • camphor and phenol
  • dolutegravir, abacavir, and lamivudine
  • peramivir
  • lisdexamfetamine
  • ergoloid mesylates
  • memantine/donepezil
  • tranylcypromine
  • isocarboxazid
  • methenamine/sodium salicylate/benzoic acid
  • mometasone topical (Rx)
  • Esketamine intranasal
  • Oracit
  • Shohls Solution
  • sodium lactate
  • sodium citrate
  • lecanemab
  • donepezil (Rx)
  • donepezil transdermal
  • sodium thiosulfate
  • ciclopirox
  • undecylenic acid
  • butenafine
  • calcium and vitamin D
  • zoledronic acid
  • calcitonin salmon
  • pizotifen
  • indoramin
  • salicylic acid acne
  • minoxidil topical
  • adapalene
  • orlistat
  • COVID-19 subunit vaccine
  • amoxicillin /vonoprazan
  • levamlodipine (Rx)
  • Omeprazole, amoxicillin, and clarithromycin
  • simvastatin/ezetimibe
  • amlodipine/atorvastatin
  • amoxicillin and clavulanate potassium
  • lansoprazole, amoxicillin, and clarithromycin
  • noradrenaline
  • carbaryl
  • botulinum toxin
  • atropine
  • artemether/lumefantrine
  • ergonovine
  • bunazosin (Not available in the United States)
  • ibalizumab
  • dolutegravir
  • hydrocodone/pseudoephedrine
  • cetirizine/pseudoephedrine
  • acetaminophen/dextromethorphan/pseudoephedrine/guaifenesin
  • acetaminophen IV/ibuprofen IV (Pending FDA Approval)
  • medroxyprogesterone
  • acetaminophen/caffeine
  • Acetaminophen/magnesium salicylate/pamabrom
  • megestrol
  • pyridoxine (vitamin B6)
  • folic acid-cyanocobalamin-pyridoxine
  • L-methylfolate-pyridoxal 5′-phosphate-methylcobalamine
  • estropipate
  • betamethasone (systemic)
  • dolutegravir and lamivudine
  • zidovudine and lamivudine
  • mineral oil (oral/rectal)
  • regular insulin
  • dextromethorphan/bupropion
  • diphenhydramine/ibuprofen
  • enfuvirtide
  • doxapram
  • methamphetamine
  • dextroamphetamine
  • ephedrine
  • brompheniramine, dextromethorphan and phenylephrine
  • aspirin, chlorpheniramine, and phenylephrine
  • acetaminophen, pheniramine, and phenylephrine
  • chlorpheniramine and phenylephrine
  • guaifenesin and phenylephrine
  • rivastigmine
  • pyridostigmine
  • arecoline
  • physostigmine
  • abobotulinumtoxinA
  • echothiophate iodide
  • malathion
  • glibenclamide
  • rimabotulinumtoxinB
  • pioglitazone
  • daxibotulinumtoxinA
  • prabotulinumtoxinA
  • mepenzolate
  • trospium
  • modafinil
  • budesonide (oral inhalation)
  • budesonide (nasal)
  • budesonide (Topical)
  • vedolizumab
  • hydrocodone and homatropine
  • homatropine (ophthalmic)
  • methscopolamine
  • oxandrolone
  • nandrolone
  • fluoxymesterone
  • procyclidine
  • biperiden
  • benztropine
  • oxymetholone
  • ipratropium
  • belladonna/opium
  • pilocarpine
  • nicotine intranasal
  • succinylcholine
  • cromolyn sodium
  • mepolizumab
  • palivizumab
  • reslizumab
  • dupilumab
  • potassium iodide
  • benzralizumab
  • beclomethasone (nasal)
  • tetrahydrozoline
  • fluticasone (topical)
  • tecovirimat
  • entacapone
  • vaccinia immune globulin intravenous (Rx)
  • smallpox (vaccinia) vaccine, live
  • terazosin
  • labetalol 
  • smallpox and monkeypox vaccine (live, nonreplicating) (US: Availability limited to health department/CDC expanded access protocol) (Rx)
  • oxymetazoline
  • xylometazoline
  • meclizine
  • prazosin
  • belinostat
  • nabilone
  • tripelennamine
  • bismuth subcitrate, metronidazole and tetracycline
  • levalbuterol
  • rifaximin
  • cotrimoxazole
  • ethacrynic acid
  • senna
  • bisacodyl
  • sodium picosulfate, citric acid, and magnesium oxide
  • kaolin
  • anastrozole
  • docusate
  • cascara
  • dichlorphenamide
  • bismuth subsalicylate
  • methylcellulose
  • magnesium sulfate 
  • talazoparib
  • diphenoxylate/atropine
  • bacillus clausii
  • psyllium
  • bifidobacterium
  • lactobacillus
  • saccharomyces boulardii
  • lanreotide
  • cyproterone
  • ramucirumab (Rx)
  • fidaxomicin
  • tobramycin (systemic)
  • dacomitinib
  • pembrolizumab
  • amikacin (systemic)
  • panitumumab
  • blinatumomab
  • durvalumab
  • olaratumab
  • necitumumab
  • moxetumomab pasudotox
  • mogamulizumab
  • inotuzumab
  • dinutuximab
  • pentamycin
  • dibekacin
  • cemiplimab
  • gemtuzumab
  • demeclocycline
  • omadacycline
  • tobramycin (ophthalmic)
  • sarecycline
  • cefiderocol
  • valrubicin
  • plicamycin
  • denileukin diftitox
  • decitabine
  • niraparib
  • methacholine
  • carbachol
  • bethanechol
  • acetylcholine
  • atezolizumab
  • raloxifene
  • avelumab
  • leucovorin
  • cladabrine
  • pralatrexate
  • meclofenamate
  • pemetrexed
  • ustekinumab
  • diroximel fumarate
  • daratumumab
  • coccidioidin skin test
  • candida albicans extract
  • brewer’s yeast
  • poliovirus vaccine, live, trivalent
  • elotuzumab
  • trimetrexate
  • l-methyl folate
  • Methyclothiazide
  • Influenza virus vaccine
  • acitretin
  • tafamidis
  • sapropterin
  • Pidotimod
  • nitisinone
  • Mipomersen
  • levetiracetam
  • Inebilizumab
  • Diethylamine salicylate
  • COVID-19 vaccine
  • Cephalothin
  • alitretinoin
  • Alitretinoin
  • methotrexate
  • Verteporfin
  • Omacetaxine
  • methyl aminolevulinate topical
  • efgartigimod alfa
  • aminolevulinic acid
  • cetuximab
  • streptozocin
  • zoster vaccine recombinant
  • lyme disease vaccine
  • human papillomavirus vaccine
  • daclizumab
  • lomustiine
  • amitriptyline
  • triptorelin
  • Tedizolid
  • rituximab
  • darolutamide
  • Altretamine
  • Varicella-zoster vaccine
  • topotecan
  • ajmaline
  • pneumococcal vaccine
  • poliovirus vaccine
  • adenovirus vaccine type 7
  • adenovirus vaccine type 4
  • brincidofovir
  • lenograstim
  • ofatumumab
  • doxorubicin
  • thioguanine
  • tetanus toxoid
  • primidone
  • lipegfilgrastim
  • pegaspargase
  • monomethyl fumarate
  • ibritumomab
  • dimethyl fumarate
  • varicella-zoster vaccine (recombinant)
  • influenza virus vaccine, h5n1, live
  • carmustine
  • influenza virus vaccine (h5n1), adjuvanted
  • influenza a (h5n1) vaccine
  • eluxadoline
  • influenza virus vaccine quadrivalent, adjuvanted
  • idecabtagene vicleucel
  • adenovirus types 4 and 7 live, oral
  • thiotepa
  • tocilizumab
  • levodopa inhaled
  • efalizumab
  • canakinumab
  • aminoglutethimide
  • ado-trastuzumab emtansine
  • adenovirus vaccine
  • zoster vaccine live
  • typhoid vaccine, live
  • influenza virus vaccine, live, trivalent
  • influenza virus vaccine, h1n1, live
  • delavirdine
  • paclitaxel
  • siltuximab
  • miconazole
  • fludarabine
  • epirubicin
  • vinblastine
  • lomustine
  • risankizumab
  • rilonacept
  • pacritinib
  • linezolid
  • griseofulvin
  • vincristine
  • rufinamide
  • phenobarbital
  • nelarabine
  • mitoxantrone
  • mitomycin
  • mitapivat
  • letermovir
  • lasmiditan
  • idarubicin
  • filgrastim
  • elagolix
  • daunorubicin
  • daclatasvir
  • carfilzomib
  • brentuximab
  • anakinra
  • alefacept
  • thalidomide
  • teriflunomide
  • rubella virus vaccine
  • ozanimod
  • mumps virus vaccine
  • measles virus vaccine
  • golimumab
  • etanercept
  • certolizumab
  • adalimumab
  • etoposide
  • mechlorethamine
  • adenovirus type 7 vaccine
  • melphalan
  • palifermin
  • pimecrolimus
  • ropeginterferon alfa 2b
  • tacrolimus
  • tofacitinib
  • amphotericin B cholesteryl sulfate
  • amphotericin B deoxycholate
  • amphotericin B liposomal
  • amphotericin B phospholipid complex
  • anthrax vaccine adsorbed
  • denosumab
  • diphtheria & tetanus toxoids
  • echinacea
  • haemophilus influenzae type b vaccine
  • hepatitis A vaccine inactivated
  • hepatitis a/b vaccine
  • hepatitis b vaccine
  • HIV vaccine
  • human papillomavirus vaccine, quadrivalent
  • hydroxyurea
  • influenza virus vaccine (H5N1)
  • influenza virus vaccine trivalent
  • influenza virus vaccine trivalent, adjuvanted
  • influenza virus vaccine trivalent, recombinant
  • meningococcal A C Y and W-135 diphtheria conjugate vaccine
  • meningococcal A C Y and W-135 polysaccharide vaccine combined
  • meningococcal group B vaccine
  • ofatumumab SC
  • pneumococcal vaccine 13-valent
  • pneumococcal vaccine heptavalent
  • pneumococcal vaccine polyvalent
  • poliovirus vaccine inactivated
  • rabies vaccine
  • sipuleucel-T
  • trastuzumab
  • trastuzumab deruxtecan
  • eslicarbazepine acetate
  • vitamin A
  • rifampin
  • belzutifan
  • belimumab
  • belatacept
  • armodafinil
  • amobarbital
  • alemtuzumab
  • ocrelizumab
  • nivolumab
  • natalizumab
  • fingolimod
  • desogestrel
  • butalbital
  • brexanolone
  • zoster vaccine
  • yellow fever vaccine
  • varicella virus vaccine
  • smallpox vaccine
  • rotavirus vaccine
  • rubella vaccine
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dicyclomine + 

glucagon

it increases the toxicity of dicyclomine

glucagon intranasal

it increases the toxicity of dicyclomine

pramlintide

pramlintide and dicyclomine increase the effect of each other through a synergistic activity

revefenacin

dicyclomine decreases the effect of revefenacin by decreasing the cholinergic transmission

secretin

dicyclomine decreases the effect of secretin by antagonistic activity

umeclidinium bromide

umeclidinium bromide and dicyclomine increase the toxicity of each other by synergism

ramosetron

anticholinergic agents increase the constipating activity of ramosetron

mianserin

it increases the anticholinergic agents

dimenhydrinate

dimenhydrinate increases the toxicity of dicyclomine due to pharmacodynamic synergism

donepezil

it decreases the effect of dicyclomine by antagonistic activity

galantamine

it decreases the effect of dicyclomine by antagonistic activity

trazodone

trazodone and dicyclomine decrease the cholinergic transmission

Actions and Spectrum: 

dicyclomine is a medication that belongs to the class of anticholinergic drugs, and it acts on the smooth muscles of the gastrointestinal (GI) tract. The actions and spectrum of dicyclomine can be summarized as follows: 

  • Antispasmodic effects: dicyclomine works by blocking the action of acetylcholine at muscarinic receptors in the smooth muscles of the GI tract, which leads to relaxation of the muscles and a decrease in spasms. This makes it useful in the treatment of conditions that involve abdominal pain and cramping, such as irritable bowel syndrome (IBS). 
  • Anti-secretory effects: dicyclomine can also reduce the secretion of gastric acid, which can be helpful in the treatment of peptic ulcers. 
  • Local anesthetic effects: dicyclomine has some local anesthetic effects on the GI tract, which can help to reduce pain and discomfort associated with GI spasms. 

The spectrum of dicyclomine includes its use in the treatment of various GI disorders, such as IBS, functional bowel disorders, diverticulitis, and peptic ulcers. dicyclomine is often used in combination with other medications, such as proton pump inhibitors (PPIs), to provide a comprehensive approach to the management of GI disorders. It is important to note that dicyclomine is a prescription medication and should only be used under the guidance of a healthcare professional. 

Frequency defined 

>10% 

Dry mouth  

Dizziness  

Blurred vision 

1-10% 

Nervousness 

Weakness 

Somnolence 

Frequency not defined 

Abdominal distension 

Confusion state 

Cycloplegia 

Delirium 

Dermatitis 

Erythema 

Fatigue 

Hallucinations 

Insomnia 

Malaise 

Palpitation 

Rash 

Syncope 

Contraindication/Caution: 

dicyclomine has several contraindications and precautions that should be considered before use. These include: 

  • Hypersensitivity: dicyclomine should not be used in patients who have a known hypersensitivity to the medication or any of its components. 
  • Glaucoma: dicyclomine should be used with caution in patients with narrow-angle glaucoma, as it can increase intraocular pressure and exacerbate the condition. 
  • Gastrointestinal obstruction: dicyclomine should not be used in patients with obstructive disorders of the GI tract, such as pyloric stenosis or paralytic ileus. 
  • Severe ulcerative colitis: dicyclomine should be used with caution in patients with severe ulcerative colitis, as it may lead to toxic megacolon. 
  • Myasthenia gravis: dicyclomine should be used with caution in patients with myasthenia gravis, as it can exacerbate muscle weakness. 
  • Children: dicyclomine should not be used in children under 6 months of age, as it can cause serious side effects. 
  • Pregnancy and breastfeeding: dicyclomine should only be used during pregnancy or breastfeeding if the potential benefits outweigh the potential risks. 

Overall, dicyclomine should be used with caution in patients with certain medical conditions and should only be used under the guidance of a healthcare professional. It is important to inform the healthcare provider of any pre-existing medical conditions or medications being taken before starting dicyclomine therapy. 

Pregnancy consideration:  

Category B 

Breastfeeding warnings: dicyclomine should not be taken by lactating females 

Pregnancy category: 

  • Category A: Satisfactory and well-controlled studies show no risk to the fetus in the first or later trimester. 
  • Category B: There is no affirmation of risk to the fetus found in animal reproduction studies, and there are not enough studies on pregnant women. 
  • Category C: Adverse effects on the fetus found with evidence in animal reproduction studies and no adequate evidence for a product in humans; Pregnant women must take care of the potential risks. 
  • Category D: There is adequate data available with sufficient evidence of human fetal risk from various platforms. However, despite potential dangers may be used only in emergency cases for potential benefits. 
  • Category X: Drugs listed in this category outweigh the risks over benefits. The drug is not for pregnant women. 
  • Category N: No data is available for the drug under this category. 

Pharmacology: 

dicyclomine is a medication that belongs to the class of anticholinergic drugs, and it works by blocking the action of acetylcholine at muscarinic receptors in the smooth muscles of the gastrointestinal (GI) tract. This leads to relaxation of the smooth muscles and a decrease in spasms, which can help to reduce abdominal pain and cramping associated with various GI disorders. 

dicyclomine is rapidly absorbed after oral administration, and it reaches peak plasma concentrations within 1 to 1.5 hours. The medication is metabolized in the liver and excreted in the urine and feces. The half-life of dicyclomine is approximately 1.5 to 2 hours, and the duration of action is 4 to 6 hours. 

In addition to its antispasmodic effects, dicyclomine also has some local anesthetic effects on the GI tract, which can help to reduce pain and discomfort associated with GI spasms. dicyclomine can also reduce the secretion of gastric acid, which can be helpful in the treatment of peptic ulcers. 

Pharmacodynamics: 

dicyclomine is an anticholinergic medication that works by blocking the action of acetylcholine at muscarinic receptors in the smooth muscles of the gastrointestinal (GI) tract. This leads to the relaxation of the smooth muscles and a decrease in spasms, which can help to reduce abdominal pain and cramping associated with various GI disorders. 

Acetylcholine is a neurotransmitter that stimulates smooth muscle contraction in the GI tract, and its effects are mediated through muscarinic receptors. dicyclomine competitively inhibits the binding of acetylcholine to muscarinic receptors, leading to reduced smooth muscle contractions and an overall decrease in GI spasms. 

In addition to its antispasmodic effects, dicyclomine also has some local anesthetic effects on the GI tract, which can help to reduce pain and discomfort associated with GI spasms. dicyclomine can also reduce the secretion of gastric acid, which can be helpful in the treatment of peptic ulcers. 

Pharmacokinetics: 

Absorption 

The bioavailability is 67% in an intramuscular injection 

The onset of action is 1-2 hours 

The duration of action is 4 hours 

The peak plasma concentration for oral is achieved in 60-90 min 

Distribution 

The volume of distribution is 3.65 L/kg 

Metabolism 

The drug gets extensively metabolized in the liver 

Elimination and Excretion 

The half-life is 1.8 hours 

The drug is excreted 80% in urine and 8% in feces

Administration: 

dicyclomine is usually taken orally, and it is available in the form of capsules, tablets, or an oral solution. The medication should be taken with water, and it can be taken with or without food. 

The dosage and frequency of dicyclomine administration depend on the specific condition being treated and the patient’s age, weight, and overall health. Typically, the recommended adult dose of dicyclomine for the treatment of functional bowel/irritable bowel syndrome is 20 mg four times daily, with the maximum dose of 40 mg four times daily. 

For children, the recommended dose of dicyclomine is based on weight and is usually lower than the adult dose. The medication should not be used in children under six months of age. 

dicyclomine should be taken as prescribed by a healthcare professional, and patients should not exceed the recommended dose or frequency of administration. It is important to follow the instructions provided by the healthcare professional and to continue taking the medication for the entire duration of the prescribed treatment. 

Patient information leaflet 

Generic Name: dicyclomine 

Pronounced: dye-SYE-kloe-meen 

Why do we use dicyclomine? 

dicyclomine is a medication that is used to treat various gastrointestinal (GI) conditions that involve spasms, cramps, and pain. It is primarily used to treat functional bowel/irritable bowel syndrome, that is characterized by abdominal pain and discomfort, bloating, and changes in bowel habits. 

In addition to functional bowel/irritable bowel syndrome, dicyclomine can also be used to treat other GI conditions, including: 

  • Gastric ulcers 
  • Gastroesophageal reflux disease (GERD) 
  • Intestinal hypermotility 
  • Colitis 
  • Pancreatitis 
  • Diverticulitis 

dicyclomine works by relaxing the smooth muscles in the GI tract, which can help to reduce spasms and pain associated with these conditions. It can also reduce the secretion of gastric acid, which can be helpful in the treatment of peptic ulcers. 

Overall, dicyclomine is a medication that acts on the smooth muscles of the GI tract to reduce spasms and pain associated with various GI disorders. It is important to note that dicyclomine is a prescription medication and should only be used under the guidance of a healthcare professional. 

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